University Lecturer
Femke Heezemans-Meijer
Department / Institute
Biomedical Engineering
Group
Recent Publications
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Femke A. Meijer,Annet O.W.M. Saris,Richard G. Doveston,Guido J.M. Oerlemans,Rens M.J.M. de Vries,Bente A. Somsen,Anke Unger,Bert Klebl,Christian Ottmann,Peter J. Cossar
Structure-Activity Relationship Studies of Trisubstituted Isoxazoles as Selective Allosteric Ligands for the Retinoic-Acid-Receptor-Related Orphan Receptor γt
Journal of Medicinal Chemistry (2021) -
Femke Anouk Meijer
Exploring Allosteric Modulation of the Nuclear Receptor RORγt from a Drug Discovery Perspective
(2021) -
Femke A. Meijer,M.C.M. van den Oetelaar,R.G. Doveston,E.N.R. Sampers,Lucas Brunsveld
Covalent Occlusion of the RORγt Ligand Binding Pocket Allows Unambiguous Targeting of an Allosteric Site
ACS Medicinal Chemistry Letters (2021) -
Femke A. Meijer,Guido J.M. Oerlemans,Luc Brunsveld
Orthosteric and Allosteric Dual Targeting of the Nuclear Receptor RORγt with a Bitopic Ligand
ACS Chemical Biology (2021) -
Rens M.J.M. de Vries,Femke A. Meijer,Richard G. Doveston,Iris A. Leijten-van de Gevel,Luc Brunsveld
Cooperativity between the orthosteric and allosteric ligand binding sites of RORγt
Proceedings of the National Academy of Sciences of the United States of America (PNAS) (2021)
Current Educational Activities
Ancillary Activities
No ancillary activities